Adrenirgic agonist part 3 epinephrine (Drug-Drug inter action , contraindication )





Adrenergic agonist part 3 (Drug-Drug  inter action , contraindication )


Drug-Drug inter action 

Digioxin : drug used in control heart beats , arrhythmia , heart failure and most symptom on heart . The mechanism gives disturbance in heart beat and blood pressure this is leading to additive effects  of epinephrine so management  should be  
avoided .

Anesthesia : especially if the drug is inhaled ( nitrous oxide , halothane … ) the mechanism gives sensitizing on heart muscle for patient , if response at high doses he might die resulting disturbance  tachycardia so the management  should be reduce doses at inhalation administration .
 
   Non selective beta blockers :  drugs used to reduce blood pressure by block beta 2 receptor so prevent agonist which  makes as vasodilator effect  of epinephrine and norepinephrine ,  but the alfa receptor not response for opposite effect . resulting increase blood pressure , the percentage of the drug in the blood increased , so the number of receptor decreased .  the management should be avoid with epinephrine .

Contraindication :

Hyperthyroidism : the epinephrine my cause hypersensitive response in thyrotoxic patient by increased of production of adrenergic beta receptor . it cause heart disease , as for recommendations it must be given by small doses and it consists partial agonist .

Diabetes mellitus :  epinephrine is help to regulate glucose in blood circulation resulting hyperglycemia . for this we will increase the dose of insulin .

The epinephrine used in emergency situation ,, gives ( intravenous ) rapid onset and duration by liver  .
When gives ( intramuscular ) and may be gives subcutaneously  to gives long t.5 .
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